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Radiolabeling of the B- and C-ring of estradiol using no-carrier-added bromine-77

✍ Scribed by Mark D. Hylarides; Alberto A. Leon; Fred A. Mettler; D. Scott Wilbur

Publisher: John Wiley and Sons
Year: 1985
Tongue: French
Weight: 316 KB
Volume: 22
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580220505

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✦ Synopsis

Two e s t r a d l o l d e r i v a t i v e s , A6and A -e s t r a d i o l 3-acetate (1) and (2) were prepared and allowed t o r e a c t u l t h Na Br and N-chlorosucclnlmlde (NCS) I n methanol. The r a p l d a d d l t l o n o f 778r-OCH3 t o t h e 8-rtng and C-rlng double bonds

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