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Protease-catalysed synthesis of Z-l-aminoacyl-l-caprolactam amides from Z-protected amino acid esters and dl-α-amino-ε-caprolactam

✍ Scribed by Alexander Lang; Peter Kuhl


Publisher
Elsevier Science
Year
2010
Tongue
French
Weight
154 KB
Volume
51
Category
Article
ISSN
0040-4039

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✦ Synopsis


The enzymatic synthesis of Z-L-aminoacyl-L-caprolactam amides from Z-protected amino acid esters and DL-a-amino-e-caprolactam (ACL) was accomplished by the thiol proteases papain, bromelain and ficin in aqueous-organic media. Product yields of 96% and 87% for Z-Gly-