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Preparation of 2,6-anhydro-3-deoxyhept-(or hex-)2-enononitriles (1-cyanoglycals) from 1-bromo-D-glycosyl cyanides with zinc under aprotic conditions

✍ Scribed by Somsák, László ;Bajza, István ;Batta, Gyula


Book ID
102366196
Publisher
John Wiley and Sons
Year
1990
Tongue
English
Weight
358 KB
Volume
1990
Category
Article
ISSN
0947-3440

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✦ Synopsis


Abstract

Acetylated 1‐bromo‐D‐glycosyl cyanides 1–5 react with zinc dust in acetic acid, acetic acid/water, or 2‐propanol to give mixtures of acetylated 1‐cyanoglycals 6–9 and anomeric pairs of glycosyl cyanides 10–14. Reaction of 1–5 in refluxing benzene in the presence of one equivalent of triethylamine or especially pyridine predominantly leads to the formation of 1‐cyanoglycals.