✦ LIBER ✦

Potent and Selective MC-4 Receptor Agonists Based on a Novel Disulfide Scaffold.

✍ Scribed by Liang Z. Yan; et al. et al.

Publisher: John Wiley and Sons
Year: 2006
Weight: 14 KB
Volume: 37
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.200602195

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Potent and Selective, Sulfamide-Based Hu

Potent and Selective, Sulfamide-Based Human β3-Adrenergic Receptor Agonists.

✍ Robert L. Dow; Ernest S. Paight; Steven R. Schneider; John R. Hadcock; Diane M. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 38 KB 👁 1 views

## Abstract For Abstract see ChemInform Abstract in Full Text.

Design of a novel pyrrolidine scaffold u

Design of a novel pyrrolidine scaffold utilized in the discovery of potent and selective human β3 adrenergic receptor agonists

✍ Gregori J. Morriello; Harvey R. Wendt; Alka Bansal; Jerry Di Salvo; Scott Feighn 📂 Article 📅 2011 🏛 Elsevier Science 🌐 English ⚖ 822 KB

A novel class of human b 3 -adrenergic receptor agonists was designed in effort to improve selectivity and metabolic stability versus previous disclosed b 3 -AR agonists. As observed, many of the b 3 -AR agonists seem to need the acyclic ethanolamine core for agonist activity. We have synthesized de

Discovery of a Novel, Potent and Selecti

Discovery of a Novel, Potent and Selective Human β3-Adrenergic Receptor Agonist.

✍ Yutaka Nakajima; Hitoshi Hamashima; Ken-Ichi Washizuka; Yasuyo Tomishima; Hiroak 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 10 KB 👁 1 views

ChemInform Abstract: Novel and Highly Po

ChemInform Abstract: Novel and Highly Potent 5-HT3 Receptor Agonists Based on a Pyrroloquinoxaline Structure.

✍ V. NACCI; ET AL. ET AL. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 35 KB 👁 2 views

Discovery of potent and selective histam

Discovery of potent and selective histamine H3 receptor inverse agonists based on the 3,4-dihydro-2H-pyrazino[1,2-a]indol-1-one scaffold

✍ H.G.F. Richter; C. Freichel; J. Huwyler; T. Nakagawa; M. Nettekoven; J.-M. Planc 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 453 KB

A novel series of potent histamine H(3) receptor inverse agonists based on the 3,4-dihydro-2H-pyrazino[1,2-a]indol-1-one scaffold has been discovered. Several compounds display high selectivity over other histamine receptor subtypes and have favorable physicochemical properties, low potential for CY

Discovery of a Potent and Selective Agon

Discovery of a Potent and Selective Agonist of the Prostaglandin EP4 Receptor.

✍ Xavier Billot; Anne Chateauneuf; Nathalie Chauret; Danielle Denis; Gillian Greig 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 70 KB 👁 2 views