Rapid throughput solubility screening me
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Jeremy Guo; Paul A. Elzinga; Michael. J. Hageman; James N. Herron
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Article
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2008
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John Wiley and Sons
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English
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A rapid solubility-screening assay was developed with a focus on Biopharmaceutic Classification Scheme (BCS) class II drug solubility in animal and simulated human gastrointestinal (GI) fluids. The assay enables biologically promising drug leads to be evaluated for solubility limitations earlier in