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Postprandial Changes in Solubilizing Capacity of Human Intestinal Fluids for BCS Class II Drugs

โœ Scribed by Sarah Clarysse; Dimitrios Psachoulias; Joachim Brouwers; Jan Tack; Pieter Annaert; Guus Duchateau; Christos Reppas; Patrick Augustijns


Book ID
106493739
Publisher
Springer US
Year
2009
Tongue
English
Weight
248 KB
Volume
26
Category
Article
ISSN
0724-8741

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Rapid throughput solubility screening me
โœ Jeremy Guo; Paul A. Elzinga; Michael. J. Hageman; James N. Herron ๐Ÿ“‚ Article ๐Ÿ“… 2008 ๐Ÿ› John Wiley and Sons ๐ŸŒ English โš– 303 KB

A rapid solubility-screening assay was developed with a focus on Biopharmaceutic Classification Scheme (BCS) class II drug solubility in animal and simulated human gastrointestinal (GI) fluids. The assay enables biologically promising drug leads to be evaluated for solubility limitations earlier in