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Piperazine-Based CCR5 Antagonists as HIV-1 Inhibitors. II. Discovery of 1-[(2,4-Dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3( S )-methyl-4-[1( S )-[4-(trifluoro- methyl)phenyl]ethyl]-1-piperazinyl]- piperidine N 1-Oxide (Sch-350634), an Orally Bioavailable, Potent CCR5 Antagonist

✍ Scribed by Tagat, Jayaram R.; Steensma, Ruo W.; McCombie, Stuart W.; Nazareno, Dennis V.; Lin, Sue-Ing; Neustadt, Bernard R.; Cox, Kathleen; Xu, Serena; Wojcik, Lisa; Murray, Michael G.; Vantuno, Nicole; Baroudy, Bahige M.; Strizki, Julie M.

Book ID: 121495707
Publisher: American Chemical Society
Year: 2001
Tongue: English
Weight: 68 KB
Volume: 44
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm0155401

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