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Phyllanthoside-Phyllanthostatin synthetic studies. 6. An augmented spiroketalization tactic for the total synthesis of phyllanthocin

✍ Scribed by Amos B. Smith III; James R. Empfield; Henry A. Vaccaro


Book ID
104212346
Publisher
Elsevier Science
Year
1989
Tongue
French
Weight
250 KB
Volume
30
Category
Article
ISSN
0040-4039

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✦ Synopsis


An enhanced spiroketalization maneuver permitting equilibration at both the C(8) and C(11) centers of spiroketals 17a,b leads to a more concise and efficient synthesis of phyllanthocin (i.e., 21 steps, 5.6% overall yield).