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Pharmacological characterization of a novel muscarinic partial agonist, YM796, in transfected cells expressing the m1 or m2 muscarinic receptor gene

✍ Scribed by Hongbing Wei; William R. Roeske; Josephine Lai; Fumikazu Wanibuchi; Kazuyuki Hidaka; Shinji Usuda; Henry I. Yamamura


Book ID
118345622
Publisher
Elsevier Science
Year
1992
Tongue
English
Weight
559 KB
Volume
50
Category
Article
ISSN
0024-3205

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Pharmacological in vitro characterizatio
✍ Eddi Meier; Kristen Frederiksen; Mogens Nielsen; Hanne LΓΈve LembΓΈl; Henrik Peder πŸ“‚ Article πŸ“… 1997 πŸ› John Wiley and Sons 🌐 English βš– 210 KB πŸ‘ 1 views

The arecoline bioisostere, Lu 25-109-T, displays a pharmacological profile of a partial muscarinic agonist with a several-fold higher affinity for cortical M 1 receptors than for brain stem M 2 receptors and salivary glands M 3 receptors. The compound is selective for muscarinic receptors as it show