𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Partial Agonists for A3 Adenosine Receptors

✍ Scribed by Zhan-Guo Gao; Kenneth A. Jacobson

Publisher
John Wiley and Sons
Year
2004
Weight
7 KB
Volume
35
Category
Article
ISSN
0931-7597

No coin nor oath required. For personal study only.

πŸ“œ SIMILAR VOLUMES

A3 adenosine receptors: Protective vs. d
A3 adenosine receptors: Protective vs. damaging effects identified using novel agonists and antagonists
✍ Kenneth A. Jacobson; Stefano Moro; Yong-Chul Kim; An-Hu Li πŸ“‚ Article πŸ“… 1998 πŸ› John Wiley and Sons 🌐 English βš– 298 KB πŸ‘ 2 views

Investigation of the physiologic role of the A 3 adenosine receptor has been facilitated by the availability of selective agonists and antagonists. Selective agonists include IB-MECA and the 2-chloro derivative Cl-IB-MECA. Selective antagonists have been identified and designed with the aid of molec

Adenosine A3 receptors and viability of
Adenosine A3 receptors and viability of astrocytes
✍ Maria P. Abbracchio; Stefania Ceruti; Roberta Brambilla; Daniela Barbieri; Aless πŸ“‚ Article πŸ“… 1998 πŸ› John Wiley and Sons 🌐 English βš– 293 KB πŸ‘ 2 views

We investigated the role of the A 3 adenosine receptor in cells of the astroglial lineage (both rat primary astrocytes and human astrocytoma ADF cells) by means of the selective A 3 agonists N 6 -(3iodobenzyl)-adenosine-5Β’-N-methyluronamide (IB-MECA) and CI-IB-MECA, and by utilizing the selective A

Agonist derived molecular probes for A2
Agonist derived molecular probes for A2 adenosine receptors
✍ Kenneth A. Jacobson; Lewis K. Pannell; Xiao-Duo Ji; Michael F. Jarvis; Michael W πŸ“‚ Article πŸ“… 1989 πŸ› John Wiley and Sons 🌐 English βš– 922 KB

The adenosine agonist 2-(4-(2-carboxyethyl)phenylethylamino)-5'-~-ethylcarboxamidoadenosine (CGS21680) was recently reported to be selective for the A, adenosine receptor subtype, which mediates its hypotensive action. To investigate structurelactivity relationships at a distal site, CGS21680 was de

ChemInform Abstract: N-Cycloalkyl Deriva
ChemInform Abstract: N-Cycloalkyl Derivatives of Adenosine and 1-Deazaadenosine as Agonists and Partial Agonists of the A1 Adenosine Receptor.
✍ Sauro Vittori; Anna Lorenzen; Christina Stannek; Stefano Costanzi; Rosaria Volpi πŸ“‚ Article πŸ“… 2010 πŸ› John Wiley and Sons βš– 32 KB πŸ‘ 1 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a β€œFull Text” option. The original article is trackable v

CoMFA Study on Adenosine A2A Receptor Ag
CoMFA Study on Adenosine A2A Receptor Agonists
✍ Doytchinova, Irini ;Valkova, Iva ;Natcheva, Roumiana πŸ“‚ Article πŸ“… 2001 πŸ› John Wiley and Sons 🌐 English βš– 205 KB πŸ‘ 2 views

A step-wise CoMFA-based procedure was applied to a series of 51 C2-oxyadenosines in order to select the most predictive conformation for binding to A 2A adenosine receptor. The highest correlation and predictive power was found for conformers with the side chain at the 2position oriented in the dire