Palladium-Catalyzed Annulation of 2-(1-Alkynyl)benzenamines with Disulfides: Synthesis of 3-Sulfenylindoles
✍ Scribed by Yan-Jin Guo; Ri-Yuan Tang; Jin-Heng Li; Ping Zhong; Xing-Guo Zhang
- Publisher
- John Wiley and Sons
- Year
- 2009
- Tongue
- English
- Weight
- 167 KB
- Volume
- 351
- Category
- Article
- ISSN
- 1615-4150
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✦ Synopsis
Abstract
3‐Sulfenylindoles can be efficiently prepared in moderate to good yields from 2‐(1‐alkynyl)benzenamines and disulfides using the palladium/air catalytic systems. The study also provides a useful route to the synthesis of fipronil analogues.
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