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Palladium-Catalyzed Alkynylation of 2-Iodo-p-carboranes and 9-Iodo-m-carboranes

โœ Scribed by I. P. Beletskaya; V. I. Bregadze; V. A. Ivushkin; G. G. Zhigareva; P. V. Petrovskii; I. B. Sivaev


Book ID
106523584
Publisher
SP MAIK Nauka/Interperiodica
Year
2005
Tongue
English
Weight
133 KB
Volume
41
Category
Article
ISSN
1070-4280

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## Abstract Many __orthoโ€/metaโ€/paraโ€closo__โ€carborane derivatives have been proposed for boron neutron capture therapy. However, it is difficult to follow their pharmacokinetics in patients, which creates a risk of suboptimal treatment. Adding a radioactive label to __closo__โ€carboranes may simpli