Opioid peptide receptor studies, 11: Inv
✍
Heng Xu; Yi-Feng Lu; John S. Partilla; Qiao-Xi Zheng; Jia-Bei Wang; George A. Br
📂
Article
📅
1999
🏛
John Wiley and Sons
🌐
English
⚖ 135 KB
👁 1 views
Previous data obtained with the cloned rat µ opioid receptor demonstrated that the ''super-potent'' opiates, ohmefentanyl (RTI-4614-4) and its four enantiomers, differ in binding affinity, potency, efficacy, and intrinsic efficacy. Molecular modeling (Tang et al., 1996) of fentanyl derivatives bindi