## Abstract A 21‐membered library of pyrimidines is prepared by the present protocol.
One-Pot Synthesis of Pyrimidines via Cyclocondensation of β-Bromovinyl Aldehydes with Amidine Hydrochlorides
✍ Scribed by Shengjiao Yan; Yajuan Tang; Fuchao Yu; Jun Lin
- Book ID
- 102256661
- Publisher
- John Wiley and Sons
- Year
- 2011
- Tongue
- German
- Weight
- 143 KB
- Volume
- 94
- Category
- Article
- ISSN
- 0018-019X
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✦ Synopsis
Abstract
A series of pyrimidines were prepared by cyclocondensation of β‐bromovinyl aldehydes with amidine hydrochlorides in the presence of Et~3~N in excellent yields (74–95%).
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