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Novel method for the preparation of monofluoroacetyl and difluoroacetylfuran derivatives

โœ Scribed by Virendra Kumar; Patrick McCloskey; Malcolm R. Bell

Book ID
104215660
Publisher
Elsevier Science
Year
1994
Tongue
French
Weight
173 KB
Volume
35
Category
Article
ISSN
0040-4039

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โœฆ Synopsis

Monofluoroacetyl and difluoroacctylsteroidal furans were prepared by selective reductive dehalogenation of chlorofluom and chlomdifluomacetyl inmm&iates with sodium formaldehyde sulfoxylate. WC have mcently qcatedl the synthesis of S-mthylsulfonyl[3,2-b]~dat fumn (1) and the androgen receptor activity of this compound. In order to explore the suuctum-activity relationship of this series of compounds, we have introduced a number of other electron withdrawing substituents at 5' position of the

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