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Mitigating hERG Inhibition: Design of Orally Bioavailable CCR5 Antagonists as Potent Inhibitors of R5 HIV-1 Replication

✍ Scribed by Skerlj, Renato; Bridger, Gary; Zhou, Yuanxi; Bourque, Elyse; McEachern, Ernest; Danthi, Sanjay; Langille, Jonathan; Harwig, Curtis; Veale, Duane; Carpenter, Bryon; Ba, Tuya; Bey, Michael; Baird, Ian; Wilson, Trevor; Metz, Markus; MacFarland, Ron; Mosi, Renee; Bodart, Veronique; Wong, Rebecca; Fricker, Simon; Huskens, Dana; Schols, Dominique

Book ID: 127388620
Publisher: American Chemical Society
Year: 2012
Tongue: English
Weight: 590 KB
Volume: 3
Category: Article
ISSN: 1948-5875
DOI: 10.1021/ml2002604

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