2-(Het)aryl-Substituted 7-Azabicyclo[2.2
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Albert Otten; Jan Christoph Namyslo; Martin Stoermer; Dieter E. Kaufmann
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Article
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1998
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John Wiley and Sons
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English
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Epibatidine (1) is a recently discovered trace alkaloid found pyrrole (7) with ethynyl p-tolyl sulfone (6) and subsequent steps has been optimized. The crucial last step, the reductive in the skin of a Latin-American poisonous frog. Its remarkably high analgetic activity is accompanied by high cleav