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Kinetic resolution of 1,1′-binaphthylamines via lipase-catalyzed amidation

✍ Scribed by Naoto Aoyagi; Taeko Izumi

Book ID
104251555
Publisher
Elsevier Science
Year
2002
Tongue
French
Weight
127 KB
Volume
43
Category
Article
ISSN
0040-4039

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✦ Synopsis

Lipase-catalyzed amidation of 2-(2-aminoethyl)-1,1%-binaphthyl (±)-3 gave optically active 2-[2-(acylamino)ethyl]-1,1%binaphthyls (R)-6a-c with high enantiomeric excess.

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