✦ LIBER ✦

Interactive SAR Studies: Rational Discovery of Super-Potent and Highly Selective Dopamine D3 Receptor Antagonists and Partial Agonists

✍ Scribed by Bettinetti, Laura; Schlotter, Karin; Hübner, Harald; Gmeiner, Peter

Book ID: 111685134
Publisher: American Chemical Society
Year: 2002
Tongue: English
Weight: 76 KB
Volume: 45
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm025558r

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and SAR of Highly Potent and S

Synthesis and SAR of Highly Potent and Selective Dopamine D3-Receptor Antagonists: 1H-Pyrimidin-2-one Derivatives.

✍ Herve Geneste; et al. et al. 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 11 KB 👁 2 views

Synthesis and SAR of Highly Potent and S

Synthesis and SAR of Highly Potent and Selective Dopamine D3-Receptor Antagonists: Quinolin(di)one and Benzazepin(di)one Derivatives.

✍ Herve Geneste; et al. et al. 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 9 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.

Synthesis and SAR of Highly Potent and S

Synthesis and SAR of Highly Potent and Selective Dopamine D3-Receptor Antagonists: Variations on the 1H-Pyrimidin-2-one Theme.

✍ Herve Geneste; et al. et al. 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 14 KB 👁 2 views

Regulation of agonist and antagonist bin

Regulation of agonist and antagonist binding to striatal D-1 dopamine receptors: Studies using the selective D-1 antagonist [3H]SK&F R-83566

✍ Kathryn E. Flaim; George W. Gessner; Stanley T. Crooke; J.Richard Heys; Joseph W 📂 Article 📅 1986 🏛 Elsevier Science 🌐 English ⚖ 624 KB

Structure–Activity Relationship Study of

Structure–Activity Relationship Study of N 6 -(2-(4-(1 H -Indol-5-yl)piperazin-1-yl)ethyl)- N 6 -propyl-4,5,6,7-tetrahydrobenzo[ d ]thiazole-2,6-diamine Analogues: Development of Highly Selective D3 Dopamine Receptor Agonists along with a Highly Potent D2/D3 Agonist and Their Pharmacological Characterization

✍ Johnson, Mark; Antonio, Tamara; Reith, Maarten E. A.; Dutta, Aloke K. 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 918 KB

The decrease of dopamine D2/D3 receptor

The decrease of dopamine D2/D3 receptor densities in the putamen and nucleus caudatus goes parallel with maintained levels of CB1 cannabinoid receptors in Parkinson's disease: A preliminary autoradiographic study with the selective dopamine D2/D3 antagonist [3H]raclopride and the novel CB1 inverse agonist [125I]SD7015

✍ Szabolcs Farkas; Katalin Nagy; Zhisheng Jia; Tibor Harkany; Miklós Palkovits; Se 📂 Article 📅 2012 🏛 Elsevier Science 🌐 English ⚖ 745 KB