✦ LIBER ✦

Interactions of inhibitor molecules with the human CYP2E1 enzyme active site

✍ Scribed by Martikainen, Laura E.; Rahnasto-Rilla, Minna; Neshybova, Silvie; Lahtela-Kakkonen, Maija; Raunio, Hannu; Juvonen, Risto O.

Book ID: 125460400
Publisher: Elsevier Science
Year: 2012
Tongue: English
Weight: 944 KB
Volume: 47
Category: Article
ISSN: 0928-0987
DOI: 10.1016/j.ejps.2012.09.018

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Inhibitor interactions with the active s

Inhibitor interactions with the active site of catechol 2,3 dioxygenase from pseudomonas putida MT2

✍ Fabrizio Briganti; Andrea Scozzafava 📂 Article 📅 1993 🏛 Elsevier Science 🌐 English ⚖ 72 KB

Activity of CYP2E1 and CYP3A enzymes in

Activity of CYP2E1 and CYP3A enzymes in adults with moderate alcohol consumption: A comparison with nonalcoholics

✍ Suthat Liangpunsakul; Dhanashri Kolwankar; Amar Pinto; J. Christopher Gorski; St 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 English ⚖ 227 KB 👁 1 views

Alcohol consumption is known to induce hepatic CYP2E1 activity, but its effect on hepatic and intestinal CYP3A in humans is not known. We have conducted a study to compare the CYP2E1 and CYP3A activities in 20 individuals with moderate alcohol consumption and 20 gender-, race-. and body mass index (

Interactions of lipoprotein lipase with

Interactions of lipoprotein lipase with the active-site inhibitor tetrahydrolipstatin (Orlistat)R

✍ Aivar LOOKENE; Nina SKOTTOVA; Gunilla OLIVECRONA 📂 Article 📅 1994 🏛 John Wiley and Sons 🌐 English ⚖ 921 KB

Discovery of Small-Molecule Inhibitors o

Discovery of Small-Molecule Inhibitors of the ATPase Activity of Human Papillomavirus E1 Helicase

✍ Faucher, Anne-Marie; White, Peter W.; Brochu, Christian; Grand-Maître, Chantal; 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 88 KB

Structure-activity relationships of sulf

Structure-activity relationships of sulfonamide drugs and human carbonic anhydrase C: Modeling of inhibitor molecules into the receptor site of the enzyme with an interactive computer graphics display

✍ Angelo Vedani; Edgar F. Meyer Jr 📂 Article 📅 1984 🏛 John Wiley and Sons 🌐 English ⚖ 702 KB

Human Cathepsin B Is a Metastable Enzyme

Human Cathepsin B Is a Metastable Enzyme Stabilized by Specific Ionic Interactions Associated with the Active Site

✍ Turk, Boris; Dolenc, Iztok; Zerovnik, Eva; Turk, Dusan; Gubensek, Franc; Turk, V 📂 Article 📅 1994 🏛 American Chemical Society 🌐 English ⚖ 813 KB