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Inhibition of rabbit lung angiotensin converting enzyme by idrapril

✍ Scribed by Annalisa Lippi; Marco Criscuoli; Giuliana Sardelli; Alessandro Subissi


Book ID
115783339
Publisher
Elsevier Science
Year
1993
Tongue
English
Weight
532 KB
Volume
45
Category
Article
ISSN
0006-2952

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Rapid reversal of angiotensin converting
✍ S. Rimar; C.N. Gillis πŸ“‚ Article πŸ“… 1992 πŸ› Elsevier 🌐 English βš– 502 KB

Lisinopril is a potent competitive inhibitor of purified rabbit lung ACE (dissociation t1/2 = 105 min). To examine reversibility of binding and ACE functional activity in situ, the single-pass extraction (E) of an 125I-lisinopril analogue (351A) and the hydrolysis of an ACE substrate, benz-phe-ala-p