Inhibition of peroxisome proliferator-activated receptor γ activity suppresses pancreatic cancer cell motility
✍ Scribed by Atsushi Nakajima; Ayako Tomimoto; Koji Fujita; Michiko Sugiyama; Hirokazu Takahashi; Ikuko Ikeda; Kunihiro Hosono; Hiroki Endo; Kyoko Yoneda; Hiroshi Iida; Masahiko Inamori; Kensuke Kubota; Satoru Saito; Noriko Nakajima; Koichiro Wada; Yoji Nagashima; Hitoshi Nakagama
- Book ID
- 108584286
- Publisher
- John Wiley and Sons
- Year
- 2008
- Tongue
- English
- Weight
- 611 KB
- Volume
- 99
- Category
- Article
- ISSN
- 1347-9032
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## Abstract BRL 49653 (rosiglitazone) is a thiazolidinedione anti‐diabetic drug that activates the nuclear receptor, peroxisome proliferator‐activated receptor gamma (PPARγ). Pilot clinical trials have shown evidence of therapeutic activity of PPARγ agonists against prostate cancer. To more effecti
## Abstract Peroxisome proliferator‐activated receptor‐gamma (PPAR‐γ) is a member of the nuclear hormone receptor superfamily of ligand‐activated transcription factors and a crucial regulator of cellular differentiation. PPAR‐γ ligands have been demonstrated to inhibit growth of several cancer cell