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Incorporation of α-trifluoromethyl substituted α-amino acids into C-and N-terminal position of peptides and peptide mimetics using multicomponent reactions

✍ Scribed by K. Burger; K. Mütze; W. Hollweck; B. Koksch

Publisher: Elsevier Science
Year: 1998
Tongue: French
Weight: 694 KB
Volume: 54
Category: Article
ISSN: 0040-4020
DOI: 10.1016/s0040-4020(98)00291-9

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✦ Synopsis

Methodology for incorporation of cz-tfifluoromethyl substituted amino acids into the Cand N-terminal position of peptides and pcptide mimcfics via multicomponcnt reactions of the Passefini and Ugi type is dcscfibed.

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