Radiolabeling of a high potency cannabin
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Sean R. Donohue; Christer Halldin; Magnus Schou; Jinsoo Hong; Lee Phebus; Eyassu
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Article
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2008
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John Wiley and Sons
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French
⚖ 216 KB
👁 1 views
## Abstract PipISB [__N__‐(4‐fluoro‐benzyl)‐4‐(3‐(piperidin‐1‐yl)‐indole‐1‐sulfonyl)benzamide, 9] was identified as a selective high potency CB~1~ receptor ligand. Here we describe the labeling of 9 with positron‐emitters to provide candidate radioligands for imaging brain CB~1~ receptors with posi