𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Heilmittelchemische Studien in der heterocyclischen Reihe. 34. Mitteilung. Pyrazolo-pyrimidine V. Eine neue Synthese von Pyrazolo[3,4-d]pyrimidinen mit coronarerweiternden Eigenschaften

✍ Scribed by P. Schmidt; K. Eichenberger; M. Wilhelm


Publisher
John Wiley and Sons
Year
1962
Tongue
German
Weight
483 KB
Volume
45
Category
Article
ISSN
0018-019X

No coin nor oath required. For personal study only.

✦ Synopsis


Abstract

Condensation of 3‐amino‐4‐carbethoxy‐pyrazoles with nitriles led to a new synthesis of 6‐C‐substituted pyrazolo[3,4‐d]pyrimidines and 6‐amino‐pyrazolo‐[3,4‐b]pyridines. The structure of the new derivatives was established by independent syntheses. The pyrazolo‐pyrimidines can be cleaved with phosphoric acid to 3‐amino‐pyrazole‐4‐carboxamide derivatives. Many of the new pyrazolo‐pyrimidines show an increase of coronary flow.