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[Handbook of Experimental Pharmacology] Phosphodiesterases as Drug Targets Volume 204 || Harnessing the Clinical Efficacy of Phosphodiesterase 4 Inhibitors in Inflammatory Lung Diseases: Dual-Selective Phosphodiesterase Inhibitors and Novel Combination Therapies

โœ Scribed by Francis, Sharron H.; Conti, Marco; Houslay, Miles D.


Book ID
115465044
Publisher
Springer Berlin Heidelberg
Year
2011
Weight
332 KB
Category
Article
ISBN
364217969X

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[Handbook of Experimental Pharmacology]
โœ Francis, Sharron H.; Conti, Marco; Houslay, Miles D. ๐Ÿ“‚ Article ๐Ÿ“… 2011 ๐Ÿ› Springer Berlin Heidelberg ๐ŸŒ German โš– 201 KB

Cyclic nucleotide phosphodiesterases (PDEs) are promising targets for pharmacological intervention. Multiple PDE genes, isoform diversity, selective expression and compartmentation of the isoforms, and an array of conformations of PDE proteins are properties that challenge development of drugs that