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From partial to full agonism: Identification of a novel 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole as a full agonist of the human GPR119 receptor

✍ Scribed by Futatsugi, Kentaro; Mascitti, Vincent; Guimarães, Cristiano R.W.; Morishita, Nao; Cai, Cuiman; DeNinno, Michael P.; Gao, Hua; Hamilton, Michael D.; Hank, Richard; Harris, Anthony R.; Kung, Daniel W.; Lavergne, Sophie Y.; Lefker, Bruce A.; Lopaze, Michael G.; McClure, Kim F.; Munchhof, Michael J.; Preville, Cathy; Robinson, Ralph P.; Wright, Stephen W.; Bonin, Paul D.; Cornelius, Peter; Chen, Yue; Kalgutkar, Amit S.

Book ID: 118148958
Publisher: Elsevier Science
Year: 2013
Tongue: English
Weight: 377 KB
Volume: 23
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2012.10.119

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