## Abstract We demonstrated the synthesis of carbon‐11 labeled 17‐__α__‐hydroxy‐11‐__β__‐/4‐/[methyl]‐[1‐methylethyl]‐aminophenyl/‐17__α__‐[prop‐1‐ynyl]esta‐4‐9‐diene‐3‐one (RU40555), a selective glucocorticoid receptor (GR) antagonist, and examined the __in vivo__ profile of [^11^C]RU40555. [^11^
✦ LIBER ✦
Evaluation of RU28318 and RU40555 as selective mineralocorticoid receptor and glucocorticoid receptor antagonists, respectively: receptor measures and functional studies
✍ Scribed by Paul J. Kim; Michael A. Cole; Brian A. Kalman; Robert L. Spencer
- Book ID
- 117669070
- Publisher
- Elsevier Science
- Year
- 1998
- Tongue
- English
- Weight
- 597 KB
- Volume
- 67
- Category
- Article
- ISSN
- 0960-0760
No coin nor oath required. For personal study only.
📜 SIMILAR VOLUMES
Synthesis and evaluation of [11C]RU40555
✍
Takahiro Matsuya; Hiroyuki Takamatsu; Yoshihiro Murakami; Akihiro Noda; Kazuhiko
📂
Article
📅
2005
🏛
John Wiley and Sons
🌐
French
⚖ 224 KB
EFFECT OF SINGLE ADMINISTRATION OF A MIN
✍
K Rahmouni; M Barthelmebs; W De Jong
📂
Article
📅
1997
🏛
John Wiley and Sons
🌐
English
⚖ 93 KB
Synthesis and Biological Evaluation of N
✍
Irini Akritopoulou-Zanze; Jyoti R. Patel; Kresna Hartandi; Jehrod Brenneman; Mar
📂
Article
📅
2004
🏛
John Wiley and Sons
⚖ 131 KB
👁 2 views
Synthesis, modification, and evaluation
✍
Cheng-Shi Jiang; Rong Zhou; Jing-Xu Gong; Li-Li Chen; Tibor Kurtán; Xu Shen; Yue
📂
Article
📅
2011
🏛
Elsevier Science
🌐
English
⚖ 385 KB
Macrolide (R)-de-O-methyllasiodiplodin (1), discovered to be a potent nonsteroidal antagonist of the mineralocorticoid receptor (MR), was synthesized via an efficient method and evaluated for MR antagonistic activity together with its analogs. Among all the tested compounds, compounds 18a, 18b and 1
Synthesis and biological evaluation of (
✍
Euna Yoo; Juhee Yoon; Ae Nim Pae; Hyewhon Rhim; Woo-Kyu Park; Jae Yang Kong; Hea
📂
Article
📅
2010
🏛
Elsevier Science
🌐
English
⚖ 367 KB
New 2-Arylpyrazolo[3,4- c ]quinoline Der
✍
Colotta, Vittoria; Catarzi, Daniela; Varano, Flavia; Capelli, Francesca; Lenzi,
📂
Article
📅
2007
🏛
American Chemical Society
🌐
English
⚖ 626 KB