Synthesis and characterization of 7α-O-i
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R. F. Wang; J. A. M. Tafani; M. Bergon; P. Tisnes; Y. Coulais; J. M. Zajac; R. G
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Article
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1995
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John Wiley and Sons
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French
⚖ 552 KB
## Abstract The preparation and synthesis of [^125^I]7α‐O‐iodoallyl diprenorphine, a high affinity opioid receptor antagonist, is described using a versatile vinylstannane as prosthetic group for radioiodination at the tertiary alcohol group in the 7α‐side chain. Radioiododestannylation with select