✦ LIBER ✦

Evaluation of [11C]SA5845 and [11C]SA4503 for imaging of sigma receptors in tumors by animal PET

✍ Scribed by Kiichi Ishiwata; Kazunori Kawamura; Kazuo Kubota; Tadayuki Kobayashi; Philip H. Elsinga; Mayumi Ono; Minoru Maeda

Publisher: Springer Japan
Year: 2005
Tongue: English
Weight: 925 KB
Volume: 19
Category: Article
ISSN: 0914-7187
DOI: 10.1007/bf02985120

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Steroid hormones affect binding of the s

Steroid hormones affect binding of the sigma ligand11C-SA4503 in tumour cells and tumour-bearing rats

✍ Anna A. Rybczynska; Philip H. Elsinga; Jurgen W. Sijbesma; Kiichi Ishiwata; Joha 📂 Article 📅 2009 🏛 Springer 🌐 English ⚖ 256 KB

Evaluation of novel PET ligands (+)N-[11

Evaluation of novel PET ligands (+)N-[11C]methyl-3-piperidyl benzilate ([11C](+)3-MPB) and its stereoisomer [11C](-)3-MPB for muscarinic cholinergic receptors in the conscious monkey brain: A PET study in comparison with [11C]4-MPB

✍ Hideo Tsukada; Kazuhiro Takahashi; Shuichi Miura; Shingo Nishiyama; Takeharu Kak 📂 Article 📅 2000 🏛 John Wiley and Sons 🌐 English ⚖ 424 KB 👁 1 views

Synthesis and biological evaluation of S

Synthesis and biological evaluation of S-[11C]methylated mercaptoimidazole piperazinyl derivatives as potential radioligands for imaging 5-HT1A receptors by positron emission tomography (PET)

✍ Raquel Garcia; Catarina Xavier; António Paulo; Isabel Santos; Torsten Kniess; R. 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 French ⚖ 157 KB

The novel 2-mercaptoimidazole derivatives, 1-[4-((2-methoxyphenyl)-1-piperazinyl)butyl]-2-mercaptoimidazole (3) and methyl[4-((2-methoxyphenyl)-1-piperazinyl))butyl] (2-mercapto-1-methylimidazol-5-yl)methanamide ( 8), were efficiently labelled with 11 C through methylation of the thioketone function

Synthesis and initial evaluation of [11C

Synthesis and initial evaluation of [11C](R)-RWAY in monkey—a new, simply labeled antagonist radioligand for imaging brain 5-HT1Areceptors with PET

✍ Julie A. McCarron; Sami S. Zoghbi; H. Umesha Shetty; Eric S. Vermeulen; Håkan V. 📂 Article 📅 2007 🏛 Springer 🌐 English ⚖ 409 KB

Synthesis of [N-methyl-11C]-3-[(6-dimeth

Synthesis of [N-methyl-11C]-3-[(6-dimethylamino)pyridin-3-yl]-2,5-dimethyl-N, N-dipropylpyrazolo[1,5-a]pyrimidine-7-amine: A potential PET ligand for in vivo imaging of CRF1 receptors

✍ J.S. Dileep Kumar; Vattoly J. Majo; Jaya Prabhakaran; Norman R. Simpson; Ronald 📂 Article 📅 2003 🏛 John Wiley and Sons 🌐 French ⚖ 138 KB

## Abstract A convenient synthesis of [N‐methyl‐^11^C]‐3‐[(6‐dimethylamino)pyridin‐3‐yl]‐2,5‐dimethyl‐__N__,__N__‐dipropylpyrazolo[1,5‐a]pyrimidine‐7‐amine (R121920), a highly selective CRF~1~ antagonist has been developed as a potential PET ligand. 3 ‐ [(6 ‐ methylamino)pyridin ‐ 3 ‐ yl]‐2,5‐dimet

Synthesis and in vivo evaluation of 3-[1

Synthesis and in vivo evaluation of 3-[11C]methyl-(3-methoxy-naphthalen)-2-yl-(1-benzyl-piperidin)-4-yl-acetate (SB-235753), as a putative dopamine D4 receptors antagonist for PET

✍ M. Matarrese; D. Soloviev; R. M. Moresco; S. Todde; P. Simonelli; D. Colombo; F. 📂 Article 📅 2000 🏛 John Wiley and Sons 🌐 French ⚖ 386 KB 👁 2 views