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Enantiospecific synthesis of the potent anti-herpetic carbocyclic 9-(2′deoxy-2′-flouro-β-D-arabinofuranosyl) guanine (+)CAFG from arsiteromycin

✍ Scribed by Alan D Borthwick; Keith Biggadike; Stuart Holman; C.L. Mo


Book ID
104226658
Publisher
Elsevier Science
Year
1990
Tongue
French
Weight
193 KB
Volume
31
Category
Article
ISSN
0040-4039

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✦ Synopsis


SlM4UZ: A ten-step enantiospecific synthesis of carkocyclic 9-(2'-deoxy-2'-fluoro-S-D-arabinofuramsyl)guanine (lo), (+) C-AEG, fran Aristerasycin is described. -We recently reported the synthesis of a new anti-herpes agent (2) carboqclic 9-(2'-deoxy-2'-flmr* p-D-arabinofuraucsyl)gua.nine (g).1,2 This fluorccarbocyclic nucleoside is highly active against Herpes Siqlex virus type 1 (HEW-l) and type 2