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Efficient chemoselective alkylation of quinoline 2,4-diol derivatives in water

✍ Scribed by Nafees Ahmed; Keyur G. Brahmbhatt; Inder P. Singh; Kamlesh K. Bhutani

Book ID: 102343076
Publisher: Journal of Heterocyclic Chemistry
Year: 2010
Tongue: English
Weight: 182 KB
Volume: 48
Category: Article
ISSN: 0022-152X
DOI: 10.1002/jhet.364

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✦ Synopsis

Abstract

Synthesis of various C‐3‐dialkyl derivatives of quinoline 2,4‐diol was achieved by condensation of aniline or substituted anilines with diethyl malonate, followed by chemoselective alkylation at C‐3 in water. The higher yields, easy work up and environmental compatible conditions are the main aspects of our method. J. Heterocyclic Chem., 2011.

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