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E. coli NfsA: an alternative nitroreductase for prodrug activation gene therapy in combination with CB1954

✍ Scribed by Vass, S O; Jarrom, D; Wilson, W R; Hyde, E I; Searle, P F


Book ID
110000061
Publisher
Nature Publishing Group
Year
2009
Tongue
English
Weight
359 KB
Volume
100
Category
Article
ISSN
0007-0920

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E. coli NfsA: an alternative nitroreduct
✍ Vass, S O; Jarrom, D; Wilson, W R; Hyde, E I; Searle, P F πŸ“‚ Article πŸ“… 2009 πŸ› Nature Publishing Group 🌐 English βš– 359 KB

Prodrug activation gene therapy is a developing approach to cancer treatment, whereby prodrug-activating enzymes are expressed in tumour cells. After administration of a non-toxic prodrug, its conversion to cytotoxic metabolites directly kills tumour cells expressing the activating enzyme, whereas t