✦ LIBER ✦

Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities

✍ Scribed by Deborah S. Kreiss; Debra A. Bergstrom; Antonio M. Gonzalez; Kai-Xing Huang; David R. Sibley; Judith R. Walters

Book ID: 115890110
Publisher: Elsevier Science
Year: 1995
Tongue: English
Weight: 497 KB
Volume: 277
Category: Article
ISSN: 0014-2999
DOI: 10.1016/0014-2999(95)00069-w

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Dopaminergic inhibition of adenylate cyc

Dopaminergic inhibition of adenylate cyclase correlates with high affinity agonist binding to anterior pituitary D2 dopamine receptors

✍ McDonald, William M.; Sibley, David R.; Kilpatrick, Brian F.; Caron, Marc G. 📂 Article 📅 1984 🏛 Elsevier Science 🌐 English ⚖ 860 KB

Affinity for Dopamine D 2 , D 3 , and D

Affinity for Dopamine D 2 , D 3 , and D 4 Receptors of 2-Aminotetralins. Relevance of D 2 Agonist Binding for Determination of Receptor Subtype Selectivity †

✍ van Vliet, L. Alexander; Tepper, Pieter G.; Dijkstra, Durk; Damsma, Geert; Wikst 📂 Article 📅 1996 🏛 American Chemical Society 🌐 English ⚖ 136 KB

Intrinsic activity of dopamine D2 agonis

Intrinsic activity of dopamine D2 agonists determined from receptor binding affinites. Correlation with in vivo activity

✍ Lahti, R.A.; Figur, L.M.; Piercey, M.F.; Ruppel, P.L.; Evans, D.L. 📂 Article 📅 1992 🏛 Elsevier Science 🌐 English ⚖ 107 KB

A novel series of arylpiperazines with h

A novel series of arylpiperazines with high affinity and selectivity for the dopamine D3 receptor

✍ P. John Murray; Lee A. Harrison; Martin R. Johnson; Graeme M. Robertson; David I 📂 Article 📅 1995 🏛 Elsevier Science 🌐 English ⚖ 210 KB

A novel series of arylpiperazines has been synthesised which show high affinity for dopamine D 3 receptors. Several of these compounds exhibit ca. 100 fold selectivity for the dopamine D 3 receptor over D 1 , D 2 and D 4 receptors. In vivo studies suggest that 4 (GR103691) may have an atypical antip

Both dopamine and the putative dopamine

Both dopamine and the putative dopamine D3 receptor antagonist PNU-99194A induce a biphasic inhibition of phorbol ester-stimulated arachidonic acid release from CHO cells transfected with the dopamine D3 receptor

✍ Christer L. Nilsson; Monika Hellstrand; Agneta Ekman; Elias Eriksson 📂 Article 📅 1999 🏛 Elsevier Science 🌐 English ⚖ 1013 KB

Characterization of binding of [3H]PD 12

Characterization of binding of [3H]PD 128907, A selective Dopamine D3 receptor agonist ligand, to CHO-K1 cells

✍ Hyacinth C. Akunne; Patrick Towers; Gareth J. Ellis; Durk Dijkstra; Håkan Wikstr 📂 Article 📅 1995 🏛 Elsevier Science 🌐 English ⚖ 772 KB