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Discovery of PF-5190457, a Potent, Selective, and Orally Bioavailable Ghrelin Receptor Inverse Agonist Clinical Candidate

✍ Scribed by Bhattacharya, Samit K.; Andrews, Kim; Beveridge, Ramsay; Cameron, Kimberly O.; Chen, Chiliu; Dunn, Matthew; Fernando, Dilinie; Gao, Hua; Hepworth, David; Jackson, V. Margaret; Khot, Vishal; Kong, Jimmy; Kosa, Rachel E.; Lapham, Kimberly; Loria, Paula M.; Londregan, Allyn T.; McClure, Kim F.; Orr, Suvi T. M.; Patel, Jigna; Rose, Colin; Saenz, James; Stock, Ingrid A.; Storer, Gregory; VanVolkenburg, Maria; Vrieze, Derek; Wang, Guoqiang; Xiao, Jun; Zhang, Yingxin

Book ID: 125515921
Publisher: American Chemical Society
Year: 2014
Tongue: English
Weight: 682 KB
Volume: 5
Category: Article
ISSN: 1948-5875
DOI: 10.1021/ml400473x

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