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Discovery of a Potent and Selective DGAT1 Inhibitor with a Piperidinyl-oxy-cyclohexanecarboxylic Acid Moiety

✍ Scribed by He, Shuwen; Hong, Qingmei; Lai, Zhong; Yang, David X.; Ting, Pauline C.; Kuethe, Jeffrey T.; Cernak, Timothy A.; Dykstra, Kevin D.; Sperbeck, Donald M.; Wu, Zhicai; Yu, Yang; Yang, Ginger X.; Jian, Tianying; Liu, Jian; Guiadeen, Deodial; Krikorian, Arto D.; Sonatore, Lisa M.; Wiltsie, Judyann; Liu, Jinqi; Gorski, Judith N.; Chung, Christine C.; Gibson, Jack T.; Lisnock, JeanMarie; Xiao, Jianying; Wolff, Michael; Tong, Sharon X.; Madeira, Maria; Karanam, Bindhu V.; Shen, Dong-Ming; Balkovec, James M.; Pinto, Shirly; Nargund, Ravi P.; DeVita, Robert J.

Book ID: 127105956
Publisher: American Chemical Society
Year: 2014
Tongue: English
Weight: 615 KB
Volume: 5
Category: Article
ISSN: 1948-5875
DOI: 10.1021/ml5003426

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