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Discovery of a novel [3.2.1] benzo fused bicyclic sulfonamide-pyrazoles as potent, selective and efficacious γ-secretase inhibitors

✍ Scribed by Ye, Xiaocong M.; Konradi, Andrei W.; Sun, Minghua; Yuan, Shendong; Aubele, Danielle L.; Dappen, Michael; Dressen, Darren; Garofalo, Albert W.; Jagodzinski, Jacek J.; Latimer, Lee; Probst, Gary D.; Sham, Hing L.; Wone, David; Xu, Ying-zi; Ness, Daniel; Brigham, Elizabeth; Kwong, Grace T.; Willtis, Chris; Tonn, George; Goldbach, Erich; Quinn, Kevin P.; Zhang, Hongbin H.; Sauer, John-Michael; Bova, Michael; Basi, Guriqbal S.

Book ID: 118233149
Publisher: Elsevier Science
Year: 2013
Tongue: English
Weight: 703 KB
Volume: 23
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2012.12.039

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