Direct conversion of 4-amino-2-oxazolines into 2-imidazolidinones
✍ Scribed by Antonio Guirado; Raquel Andreu; Jesús Gálvez
- Publisher
- Elsevier Science
- Year
- 1999
- Tongue
- French
- Weight
- 154 KB
- Volume
- 40
- Category
- Article
- ISSN
- 0040-4039
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✦ Synopsis
A convenient new method for the synthesis of polysubstituted 2-imidazolidinones has been established involving the reaction of 4-alkylamino-2-aryl-2-oxazolines with arylsulfonyl isocyanates. It has been applied successfully in preparing previously unknown 3-alkyl-4-aroylamino-l-arylsulfonyl-2-imidazolidinones in high yields.
📜 SIMILAR VOLUMES
A novel heterocycle-heterocycle inter-conversion is reported. It enables direct and efficient syntheses of either polysubstituted 2-arylimino-1,3-oxazolidine or 2-arylimino-1,3-thiazolidine hydrochlorides by a one-pot treatment of 4-amino-2phenyl-2-oxazolines with arylisocyanates or arylisothiocyana