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Dibasic Benzo[ b ]thiophene Derivatives as a Novel Class of Active Site-Directed Thrombin Inhibitors. 1. Determination of the Serine Protease Selectivity, Structure−Activity Relationships, and Binding Orientation

✍ Scribed by Sall, Daniel J.; Bastian, Jolie A.; Briggs, Stephen L.; Buben, John A.; Chirgadze, Nickolay Y.; Clawson, David K.; Denney, Michael L.; Giera, Deborah D.; Gifford-Moore, Donetta S.; Harper, Richard W.; Hauser, Kenneth L.; Klimkowski, Valentine J.; Kohn, Todd J.; Lin, Ho-Shen; McCowan, Jefferson R.; Palkowitz, Alan D.; Smith, Gerald F.; Takeuchi, Kumiko; Thrasher, Kenneth J.; Tinsley, Jennifer M.; Utterback, Barbara G.; Yan, Sau-Chi B.; Zhang, Minsheng

Book ID: 125932109
Publisher: American Chemical Society
Year: 1997
Tongue: English
Weight: 243 KB
Volume: 40
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm9704107

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