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Diastereoselective alkylation of acetoacetates of chiral inductors. Synthetic applications

✍ Scribed by N. Gálvez; M. Moreno-Mañas; R. M. Sebastián; N. Serra; E. Trepat; A. Vallribera; E. Molins

Publisher
Journal of Heterocyclic Chemistry
Year
2000
Tongue
English
Weight
686 KB
Volume
37
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

Diastereoselective alkylations of acetoacetates of chiral inductors are reviewed. The formed products are starting materials for the preparation of enantiomerically pure amino acids, 4,4‐disub‐stituted 2‐pyrazolin‐5‐ones, and of oxazoles and pyrazoles incorporating the chiral inductors.

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