Development of a Suzuki Cross-Coupling Reaction between 2-Azidoarylboronic Pinacolate Esters and Vinyl Triflates To Enable the Synthesis of [2,3]-Fused Indole Heterocycles

Fundamentals of Early Clinical Drug Deve

Fundamentals of Early Clinical Drug Development (From Synthesis Design to Formulation) || Development and Scale-Up of a Heterocyclic Cross-Coupling for the Synthesis of 5-[2-(3-Methyl-3 H -imidazol-4-yl)-thieno[3,2- b ]pyridine-7-yl] amino-2-methyl-1 H -indole

✍ Abdel-Magid, Ahmed F.; Caron, Stéphane 📂 Article 📅 2006 🏛 John Wiley & Sons, Inc. 🌐 English ⚖ 376 KB

Using Recent Examples And Important Case Studies, The Fundamentals Of Early Clinical Drug Development: From Synthesis Design To Formulation Demonstrates The Central Role℗¡that Organic Synthesis Plays In The Early Clinical Evaluation Of Potential Drug Candidates. Reflections On Process Research Ii /