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Deuteration of acetanilides and other substituted aromatics using [Ir(COD)(Cy3P)(Py)]PF6 as catalyst

✍ Scribed by D. Hesk; P. R. Das; B. Evans


Publisher
John Wiley and Sons
Year
1995
Tongue
French
Weight
295 KB
Volume
36
Category
Article
ISSN
0022-2135

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✦ Synopsis


Deuterium exchange labelling using [Ir(COD)(Cy3P)(Py)]PFg as catalyst and deuterium gas was studied on a number of substituted acetanilides. In most cases products containing deuterium ortlio to the anilide group were obtained with a high degree of enrichment. With one exception no evidence for nietn, p r n or anilide methyl labelling was seen. The catalyst was also effective in the ortlia deuteration of acetophenone, benzophenone and the P-lactam containing compound Sch 48461.