## Abstract Twenty analogues were synthesized of [Pmp^1^, D‐Trp^2^, Arg^8^]oxytocin, PA, (Pmp = β,β‐pentamethylene‐β‐mercaptopropionic acid), a potent antagonist of the uterotonic effect of oxytocin in the rat (uterotonic test __in vitro__, pA~2~ = 7.77) and in the baboon. Systematic substitution o
✦ LIBER ✦
Design of potent oxytocin antagonists featuring D-tryptophan at position 2
✍ Scribed by Flouret, George; Brieher, William; Mahan, Kevin; Wilson, Laird
- Book ID
- 126895279
- Publisher
- American Chemical Society
- Year
- 1991
- Tongue
- English
- Weight
- 740 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0022-2623
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