## Abstract The synthesis of the novel pentagastrin seco‐CBI conjugate **3**, which is based on the highly cytotoxic antitumor antibiotic (+)‐duocarmycin SA (**1**), is reported. A key step in the synthesis is the palladium‐catalyzed carbonylation of aryl bromide **7** to give the benzyl ester **16
Design and Synthesis of a PSMA Inhibitor–Doxorubicin Conjugate for Targeted Prostate Cancer Therapy
✍ Scribed by Sarva Jayaprakash; Xinning Wang; Warren D. Heston; Alan P. Kozikowski
- Publisher
- John Wiley and Sons
- Year
- 2006
- Tongue
- English
- Weight
- 208 KB
- Volume
- 1
- Category
- Article
- ISSN
- 1860-7179
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