✦ LIBER ✦

Design and syntheses of melanocortin subtype-4 receptor agonists. Part 2: Discovery of the dihydropyridazinone motif

✍ Scribed by Feroze Ujjainwalla; Daniel Warner; Christine Snedden; Ricky D. Grisson; Thomas F. Walsh; Matthew J. Wyvratt; Rubana N. Kalyani; Tanya MacNeil; Rui Tang; David H. Weinberg; Lex Van der Ploeg; Mark T. Goulet

Book ID: 108073714
Publisher: Elsevier Science
Year: 2005
Tongue: English
Weight: 717 KB
Volume: 15
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2005.06.033

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Design and Syntheses of Melanocortin Sub

Design and Syntheses of Melanocortin Subtype-4 Receptor Agonists: Evolution of the Pyridazinone Archetype.

✍ Feroze Ujjainwalla; et al. et al. 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 141 KB

Design and syntheses of melanocortin sub

Design and syntheses of melanocortin subtype-4 receptor agonists: evolution of the pyridazinone archetype

✍ Feroze Ujjainwalla; Daniel Warner; Thomas F. Walsh; Matthew J. Wyvratt; Changyou 📂 Article 📅 2003 🏛 Elsevier Science 🌐 English ⚖ 220 KB

Synthesis and Structure−Activity Relatio

Synthesis and Structure−Activity Relationships of Novel Arylpiperazines as Potent and Selective Agonists of the Melanocortin Subtype-4 Receptor

✍ Richardson, Timothy I.; Ornstein, Paul L.; Briner, Karin; Fisher, Matthew J.; Ba 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 209 KB

Discovery of Prototype Peptidomimetic Ag

Discovery of Prototype Peptidomimetic Agonists at the Human Melanocortin Receptors MC1R and MC4R

✍ Haskell-Luevano, Carrie; Hendrata, Siska; North, Cheryl; Sawyer, Tomi K.; Hadley 📂 Article 📅 1997 🏛 American Chemical Society 🌐 English ⚖ 214 KB

Discovery of (2S)-N-[(1R)-2-[4-cyclohexy

Discovery of (2S)-N-[(1R)-2-[4-cyclohexyl-4-[ [(1,1-dimethylethyl)-amino]carbonyl]-1-piperidinyl]-1- [(4-fluorophenyl)methyl]-2-oxoethyl]-4-methyl-2-piperazinecarboxamide (MB243) (I), a Potent and Selective Melanocortin Subtype-4 Receptor Agonist.

✍ Brenda L. Palucki; et al. et al. 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 10 KB 👁 1 views

Stereochemical Studies of the Monocyclic

Stereochemical Studies of the Monocyclic Agouti-Related Protein (103−122) Arg-Phe-Phe Residues: Conversion of a Melanocortin-4 Receptor Antagonist into an Agonist and Results in the Discovery of a Potent and Selective Melanocortin-1 Agonist

✍ Joseph, Christine G.; Wang, Xiang S.; Scott, Joseph W.; Bauzo, Rayna M.; Xiang, 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 202 KB