✦ LIBER ✦

Design and Microwave-Assisted Synthesis of Novel Macrocyclic Peptides Active at Melanocortin Receptors: Discovery of Potent and Selective hMC5R Receptor Antagonists

✍ Scribed by Grieco, Paolo; Cai, Minying; Liu, Lu; Mayorov, Alexander; Chandler, Kevin; Trivedi, Dev; Lin, Guangxin; Campiglia, Pietro; Novellino, Ettore; Hruby, Victor J.

Book ID: 124162807
Publisher: American Chemical Society
Year: 2008
Tongue: English
Weight: 930 KB
Volume: 51
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm701181n

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Structure−Activity Relationships of γ-MS

Structure−Activity Relationships of γ-MSH Analogues at the Human Melanocortin MC3, MC4, and MC5 Receptors. Discovery of Highly Selective hMC3R, hMC4R, and hMC5R Analogues

✍ Balse-Srinivasan, Preeti; Grieco, Paolo; Cai, Minying; Trivedi, Dev; Hruby, Vict 📂 Article 📅 2003 🏛 American Chemical Society 🌐 English ⚖ 78 KB

Structure−Activity Studies of the Melano

Structure−Activity Studies of the Melanocortin Peptides: Discovery of Potent and Selective Affinity Antagonists for the h MC3 and h MC4 Receptors †

✍ Grieco, Paolo; Lavecchia, Antonio; Cai, Minying; Trivedi, Devendra; Weinberg, Da 📂 Article 📅 2002 🏛 American Chemical Society 🌐 English ⚖ 131 KB

ChemInform Abstract: Design and Synthesi

ChemInform Abstract: Design and Synthesis of a Novel Class of Highly Potent Selective and Orally Active Non-peptide Bradykinin B2 Receptor Antagonists

✍ Hiroshi Kayakiri; Yoshito Abe; Teruo Oku 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 26 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

Synthesis and structure-activity relatio

Synthesis and structure-activity relationships of a novel series of non-peptide AT2-selective angiotensin II receptor antagonists

✍ M.T. Wu; T.J. Ikeler; W.T. Ashton; R.S.L. Chang; V.J. Lotti; W.J. Greenlee 📂 Article 📅 1993 🏛 Elsevier Science 🌐 English ⚖ 443 KB

Design, Synthesis, and Structure−Activit

Design, Synthesis, and Structure−Activity Relationships of Phthalimide-Phenylpiperazines: A Novel Series of Potent and Selective α1a-Adrenergic Receptor Antagonists

✍ Kuo, Gee-Hong; Prouty, Catherine; Murray, William V.; Pulito, Virginia; Jolliffe 📂 Article 📅 2000 🏛 American Chemical Society 🌐 English ⚖ 222 KB

Potent and Selective Peptide Agonists of

Potent and Selective Peptide Agonists of α-Melanocyte Stimulating Hormone (αMSH) Action at Human Melanocortin Receptor 5; their Synthesis and Biological Evaluation in vitro

✍ Maria A. Bednarek; Tanya MacNeil; Rui Tang; Tung M. Fong; M. Angeles Cabello; Ma 📂 Article 📅 2007 🏛 John Wiley and Sons 🌐 English ⚖ 168 KB