## Abstract An extension of the __cyclo__Sal‐pronucleotide approach is presented. Attachment of an enzyme‐cleavable ester/acylal group to the __cyclo__Sal‐d4TMP triesters should allow these compounds to be trapped intracellularly after cleavage. The ester/acylal groups were introduced in the 3‐ or
✦ LIBER ✦
d4TMP Delivery from 7-Substituted cycloSal-d4TMPs
✍ Scribed by C. Meier; J. T. Renze; J. Balzarini; E. De Clercq
- Publisher
- John Wiley and Sons
- Year
- 2004
- Weight
- 51 KB
- Volume
- 35
- Category
- Article
- ISSN
- 0931-7597
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