High yield synthesis of 4H-1,4-benzothia
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Stefania De Montis; Claudia Fattuoni; Enzo Cadoni; Maria G. Cabiddu; Michele Usa
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Article
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2008
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Journal of Heterocyclic Chemistry
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English
β 355 KB
## Abstract magnified image 4__H__β1,4βBenzothiazineβ1,1βdioxide derivatives were synthesized through a sequence of almost quantitative reactions. The commercial starting material 2β(methylsulfanyl)aniline was Bocβprotected, __N__βacylated and oxidized at the sulfur atom to obtain a sulfonyl deriv