✦ LIBER ✦

Conformationally Constrained 1,3-Diamino Ketones: A Series of Potent Inhibitors of the Cysteine Protease Cathepsin K

✍ Scribed by Marquis, Robert W.; Yamashita, Dennis S.; Ru, Yu; LoCastro, Stephen M.; Oh, Hye-Ja; Erhard, Karl F.; DesJarlais, Renee L.; Head, Martha S.; Smith, Ward W.; Zhao, Baoguang; Janson, Cheryl A.; Abdel-Meguid, Sherin S.; Tomaszek, Thaddeus A.; Levy, Mark A.; Veber, Daniel F.

Book ID: 120647098
Publisher: American Chemical Society
Year: 1998
Tongue: English
Weight: 191 KB
Volume: 41
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm980295f

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Design of Potent, Selective, and Orally

Design of Potent, Selective, and Orally Bioavailable Inhibitors of Cysteine Protease Cathepsin K

✍ Tavares, Francis X.; Boncek, Virginia; Deaton, David N.; Hassell, Anne M.; Long, 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 381 KB

Cyclic Ketone Inhibitors of the Cysteine

Cyclic Ketone Inhibitors of the Cysteine Protease Cathepsin K

✍ Marquis, Robert W.; Ru, Yu; Zeng, Jin; Trout, Robert E. Lee; LoCastro, Stephen M 📂 Article 📅 2001 🏛 American Chemical Society 🌐 English ⚖ 293 KB

2-Cyano-pyrimidines: A New Chemotype for

2-Cyano-pyrimidines: A New Chemotype for Inhibitors of the Cysteine Protease Cathepsin K

✍ Altmann, Eva; Aichholz, Reiner; Betschart, Claudia; Buhl, Thomas; Green, Jonatha 📂 Article 📅 2007 🏛 American Chemical Society 🌐 English ⚖ 180 KB

Solid-Phase Synthesis of a Combinatorial

Solid-Phase Synthesis of a Combinatorial Array of 1,3-Bis(acylamino)-2-butanones, Inhibitors of the Cysteine Proteases Cathepsins K and L

✍ Yamashita, Dennis S.; Dong, Xiaoyang; Oh, Hye-Ja; Brook, Christopher S.; Tomasze 📂 Article 📅 1999 🏛 American Chemical Society 🌐 English ⚖ 196 KB

3,4-Disubstituted Azetidinones as Select

3,4-Disubstituted Azetidinones as Selective Inhibitors of the Cysteine Protease Cathepsin K. Exploring P3 Elements for Potency and Selectivity.

✍ Eduardo L. Setti; Dana Davis; James W. Janc; Douglas A. Jeffery; Harry Cheung; W 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 11 KB 👁 2 views