The 2-(1,2-dihydro-3-oxo-3H-pyrazol-2-yl)benzothiazole scaffold was selected as a central core structure for the discovery of novel antibacterial compounds. A systematic variation of the substituents on the oxo-pyrazole moiety, as well as on the benzo moiety, led to the creation of a small and focus
✦ LIBER ✦
Conformation and ortho steric effects in a series of 2-(pyrazol-1-yl)quinolines
✍ Scribed by Shiv P. Singh; Dalip Kumar; Devinder Kumar; Ana Martínez; José Elguero
- Book ID
- 112131472
- Publisher
- Journal of Heterocyclic Chemistry
- Year
- 1996
- Tongue
- English
- Weight
- 296 KB
- Volume
- 33
- Category
- Article
- ISSN
- 0022-152X
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