𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Condensed 1,2,4-Triazines I: Behaviour of Phenanthro[9,10-e]-1,2,4-triazine Derivatives Towards Alkylating and Reducing Agends, Grignard Reagents, and Amines

✍ Scribed by Mohamed Mohamed Mohamed Sallam; Yehia Abdu Ibrahim; Sayed Abdel-Latif Abdel-Hady


Publisher
John Wiley and Sons
Year
1976
Tongue
German
Weight
372 KB
Volume
59
Category
Article
ISSN
0018-019X

No coin nor oath required. For personal study only.

✦ Synopsis


Abstract

Alkylation of 3‐hydroxy‐phenanthro[9,10‐e]1,2,4‐triazine (1a) yielded the N(2)‐alkyl derivatives 2a2b; alkylation of the 3‐mercapto analogue 1b yielded the S‐alkyl derivatives 1f1i.

1a1b reacted with alkyl and aralkylmagnesium halides to yield the corresponding 3‐hydroxy‐, and 3‐mercapto‐5‐alkyl‐(aralkyl)‐phenanthro[9,10‐e]2,3,4,5‐tetrahydro‐1,2,4‐triazines 5a5f.

Reduction of 1a yielded the hexahydrotriazine derivative 7. Amination of 1c yielded the 3‐amino derivatives 1j1o after prolonged heating.